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MediCaine MEDICAINE
THE SCIENCE

ENGINEERED TO DOMINATE

Multi-agent synergy for faster onset, deeper penetration, and longer duration. Understanding why MediCaine outperforms single-agent numbing.

WHY MULTI-AGENT?

Single-agent topical anesthetics rely on one pathway to block pain. MediCaine uses multiple agents that attack pain signals through different mechanisms simultaneously — surface blockade, deep tissue penetration, extended duration, and vascular constriction.

The result: faster onset, deeper numbing, longer duration, and reduced bleeding at the treatment site. Each agent amplifies the others through pharmaceutical synergy.

15
Min Onset
5
Hr Duration
4
Agents Max
MediCaine pharmacist
ACTIVE AGENTS

THE INGREDIENTS

Five pharmaceutical agents, each with a specific role in the numbing cascade.

B

BENZOCAINE 20%

Ester-type local anesthetic that provides rapid surface-level numbing. Blocks sodium channels on contact for immediate relief at the application site. The fastest-acting agent in the BLT formula.

Rapid Onset Surface Blockade Pro & Ultra
L

LIDOCAINE 10-30%

The gold standard of local anesthetics. Amide-type anesthetic that penetrates deep tissue layers, delivering reliable, long-lasting numbness. Present in all three MediCaine tiers at varying concentrations — 10% in Pro and Ultra, 30% in Elite.

Deep Penetration Long-Lasting All Strengths
T

TETRACAINE 7-10%

Long-duration ester anesthetic with an extended half-life. Enhances depth of nerve block and extends the numbing window significantly beyond what Lidocaine alone achieves. 10% in Pro and Ultra, 7% in Elite.

Extended Duration Deep Nerve Block All Strengths
P

PRILOCAINE 8%

Fourth-agent amplifier exclusive to the Ultra. Amide anesthetic that works synergistically with the BLT base to achieve maximum potency across all tissue depths. Adds a fourth pathway for comprehensive pain signal blockade.

Synergistic Amplifier Maximum Potency Ultra Only
Ph

PHENYLEPHRINE 0.5%

Vasoconstrictor that localizes the anesthetic effect. Constricts blood vessels at the treatment site to reduce bleeding, keep the anesthetic agents concentrated in the target area longer, and extend overall duration.

Vasoconstrictor Reduces Bleeding Pro & Ultra
COMPARISON

MEDICAINE VS INDUSTRY STANDARD

MEDICAINE
15-25 minute onset
Up to 5 hours duration
Multi-agent synergy (up to 4 anesthetics)
Vasoconstrictor reduces bleeding
Compounded fresh per order
Airless pump option for zero waste
TYPICAL NUMBING
30-45 minute onset
1-2 hours duration
Single-agent formula (Lidocaine only)
No vasoconstrictor
Mass-manufactured, long shelf sits
Jar-only, no dosing precision

READY TO ORDER?

Experience the science behind better numbing. Compounded fresh per order in the USA.